Mark Burlingame, PhD
Instrumentation Facility Mgr
Pharmaceutical Chemistry
School of Pharmacy

Publications (14)

Top publication keywords:
BacteriocinsArylsulfonatesBacillus subtilisSchistosomicidesAlkanesLactonesStaphylococcaceaeMotilinDisulfidesCarbamatesPyronesProdrugsErythromycinSchistosoma mansoniProteins

• TPT sulfonate, a single, oral dose schistosomicidal prodrug: In vivo efficacy, disposition and metabolic profiling.
  International journal for parasitology. Drugs and drug resistance 2018 Wolfe AR, Neitz RJ, Burlingame M, Suzuki BM, Lim KC, Scheideler M, Nelson DL, Benet LZ, Caffrey CR
• Identification and Optimization of Thienopyridine Carboxamides as Inhibitors of HIV Regulatory Complexes.
  Antimicrobial agents and chemotherapy 2017 Nakamura RL, Burlingame MA, Yang S, Crosby DC, Talbot DJ, Chui K, Frankel AD, Renslo AR
• Capture of micrococcin biosynthetic intermediates reveals C-terminal processing as an obligatory step for in vivo maturation.
  Proceedings of the National Academy of Sciences of the United States of America 2016 Bewley KD, Bennallack PR, Burlingame MA, Robison RA, Griffitts JS, Miller SM
• Reconstitution and Minimization of a Micrococcin Biosynthetic Pathway in Bacillus subtilis.
  Journal of bacteriology 2016 Bennallack PR, Bewley KD, Burlingame MA, Robison RA, Miller SM, Griffitts JS
• Simple one-pot synthesis of disulfide fragments for use in disulfide-exchange screening.
  ACS combinatorial science 2011 Burlingame MA, Tom CT, Renslo AR

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• Turning a protein kinase on or off from a single allosteric site via disulfide trapping.
  Proceedings of the National Academy of Sciences of the United States of America 2011 Sadowsky JD, Burlingame MA, Wolan DW, McClendon CL, Jacobson MP, Wells JA
• Structure-activity relationships of 9-substituted-9-dihydroerythromycin-based motilin agonists: optimizing for potency and safety.
  Journal of medicinal chemistry 2009 Shaw SJ, Chen Y, Zheng H, Fu H, Burlingame MA, Marquez S, Li Y, Claypool M, Carreras CW, Crumb W, Hardy DJ, Myles DC, Liu Y
• Preparation of erythromycin analogs having functional groups at C-15.
  The Journal of antibiotics 2006 Ashley GW, Burlingame M, Desai R, Fu H, Leaf T, Licari PJ, Tran C, Abbanat D, Bush K, Macielag M
• A series of 23,24-dihydrodiscodermolide analogues with simplified lactone regions.
  Bioorganic & medicinal chemistry letters 2006 Shaw SJ, Sundermann KF, Burlingame MA, Zhang D, Petryka J, Myles DC
• Toward understanding how the lactone moiety of discodermolide affects activity.
  Journal of the American Chemical Society 2005 Shaw SJ, Sundermann KF, Burlingame MA, Myles DC, Freeze BS, Xian M, Brouard I, Smith AB
• Design, synthesis, and evaluation of analogues of (+)-14-normethyldiscodermolide.
  Organic letters 2005 Smith AB, Freeze BS, Lamarche MJ, Hirose T, Brouard I, Xian M, Sundermann KF, Shaw SJ, Burlingame MA, Horwitz SB, Myles DC
• Design, synthesis, and evaluation of carbamate-substituted analogues of (+)-discodermolide.
  Organic letters 2005 Smith AB, Freeze BS, Lamarche MJ, Hirose T, Brouard I, Rucker PV, Xian M, Sundermann KF, Shaw SJ, Burlingame MA, Horwitz SB, Myles DC
• Design, synthesis and cytotoxicity of 7-deoxy aryl discodermolide analogues.
  Bioorganic & medicinal chemistry letters 2004 Burlingame MA, Shaw SJ, Sundermann KF, Zhang D, Petryka J, Mendoza E, Liu F, Myles DC, LaMarche MJ, Hirose T, Scott Freeze B, Smith AB
• Saccharopolyspora erythraea-catalyzed bioconversion of 6-deoxyerythronolide B analogs for production of novel erythromycins.
  Journal of biotechnology 2002 Carreras C, Frykman S, Ou S, Cadapan L, Zavala S, Woo E, Leaf T, Carney J, Burlingame M, Patel S, Ashley G, Licari P